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Exelixis Inc Patents

What Exelixis Inc has filed at the patent office — applications as well as grants, because a filing is on the record eighteen months before anyone has to say what it was for.

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Filings on file
54
Granted
3
Still pending
51
Filed under
2 names

54 filings

Newest filing first. A pending application has no patent number yet, and most never get one.

InventionPatent
ANTIBODY-DRUG CONJUGATES AND METHODS OF THEIR USEFiled as EXELIXIS, INC.2026-03-20AMY PETERSONpending
5T4 ANTIBODY DRUG CONJUGATES AND METHODS OF THEIR USEFiled as EXELIXIS, INC.2026-03-06AMY PETERSONpending
Processes for Preparing Quinoline Compounds and Pharmaceutical Compositions Containing Such CompoundsA61P 35/00, A61K 31/47, C07D 215/22, C07D 215/233Filed as Exelixis, Inc.2026-02-11Jo Ann Wilsonpending
FUSED PYRAZOLE DERIVATIVES AS USP1 INHIBITORSFiled as EXELIXIS, INC.2026-01-06Chandrasekhar Abbinenipending
PROCESSES FOR PREPARING QUINOLINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH COMPOUNDSFiled as Exelixis, Inc.2025-12-12Jo Ann Wilsonpending
DLL3 ANTIBODY-DRUG CONJUGATES AND USES THEREOFFiled as EXELIXIS, INC.2025-09-16Kathleen GOGASpending
C-Met Modulator Pharmaceutical CompositionsA61K 31/47, A61K 9/00, A61K 9/2004, A61K 9/2009, A61K 9/2013, A61K 9/2018, A61K 9/2031, A61K 9/2054, A61K 9/2095, A61K 9/28, A61K 9/2833, A61K 9/2866, A61K 9/2893, A61K 31/00, A61K 31/33, A61K 31/395, A61K 31/435, A61K 45/06Filed as Exelixis, Inc.2025-08-20Jo Ann Wilsonpending
METHODS OF USE OF AGENTS THAT BIND TO NKG2A AND PD-L1Filed as EXELIXIS, INC.2025-07-30SEEMA KANTAKpending
AGENTS THAT BIND TO NKG2A AND PD-L1 AND USES THEREOFA61P 29/00, C07K 16/2803, C07K 16/2827, A61P 37/00, A61P 37/04, A61P 35/00, A61K2039/505, C07K2317/31, C07K2317/32, C07K2317/33, C07K2317/34, C07K2317/515, C07K2317/522, C07K2317/524, C07K2317/526, C07K2317/565, C07K2317/567, C07K2317/73, C07K2317/75, C07K2317/76, C07K2317/92Filed as EXELIXIS, INC.2025-07-25Bonnie HAMMERpending
NKG2A BINDING AGENTS AND USES THEREOFA61P 35/00, C07K 16/2803, A61K 47/6849, A61P 37/00, A61K2039/505, C07K2317/24, C07K2317/30, C07K2317/31, C07K2317/34, C07K2317/565, C07K2317/567, C07K2317/76, C07K2317/92Filed as EXELIXIS, INC.2025-07-25Bonnie HAMMERpending
COMPOUNDS THAT INHIBIT PKMYT1A61K 31/437, C07D 471/04, A61K 31/404, A61K 31/416, A61K 31/4184, A61K 31/4192, A61K 31/444, C07D 209/42, C07D 231/56, C07D 235/06, C07D 235/08, C07D 235/10, C07D 249/18, C07D 401/04Filed as Exelixis, Inc.2025-06-18Wei Xupending
Compounds that Inhibit PKMYT1C07D 401/04, C07D 471/04, A61P 35/00, A61K 31/4375, A61K 31/444, A61K 31/47, A61K 31/4709, A61K 31/472, A61K 31/498, A61K 31/4985, A61K 31/501, A61K 31/506, A61K 31/517, A61K 31/519, A61K 31/5377, C07D 215/48, C07D 215/50, C07D 217/02, C07D 217/24, C07D 241/42, C07D 241/44, C07D 403/04, C07D 413/04, C07D 417/04, C07D 487/04, C07D 491/107, C07D 519/00Filed as Exelixis, Inc.2025-05-23Wei XUpending
PROCESSES FOR PREPARING QUINOLINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH COMPOUNDSA61P 35/00, A61K 31/47, C07D 215/22, C07D 215/233Filed as Exelixis, Inc.2025-05-08Jo Ann Wilsonpending
SOMATOSTATIN RECEPTOR 2 AGONISTS AND USES THEREOFA61K 31/4745, C07D 213/78, C07D 215/233, A61P 3/10, A61K 31/4436, A61K 31/444, A61K 31/47, A61K 31/4709, A61K 31/496, A61K 31/519, C07D 213/74, C07D 215/12, C07D 401/04, C07D 401/14, C07D 471/04, C07D 471/10, C07D 471/14, C07D 471/18, C07D 471/22, C07D 487/10, C07D 491/048, C07D 491/052, C07D 491/08, C07D 495/04, C07D 498/18, C07D 513/16, C07D 513/22Filed as Exelixis, Inc.2025-04-25Dongcheng DAIpending
4,5,6,7-TETRAHYDRO-1H-PYRAZOLO[4,3-c]PYRIDINE COMPOUNDS AND DERIVATIVES AS USP1 INHIBITORSC07D 471/04, A61P 35/00, A61K 31/437, A61K 31/444, A61K 31/506Filed as EXELIXIS, INC.2025-04-18Chandrasekhar ABBINENIpending
ANTIBODY-DRUG CONJUGATES AND METHODS OF THEIR USEFiled as EXELIXIS, INC.2025-03-21Amy PETERSONpending
5T4 ANTIBODY DRUG CONJUGATES AND METHODS OF THEIR USEFiled as EXELIXIS, INC.2025-03-07Amy PETERSONpending
Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms thereof for the treatment of cancerC07D 215/22, C07D 215/233, A61K 31/47, A61P 43/00, A61P 25/00, A61P 5/14, A61P 35/00, C07B2200/13Filed as Exelixis, Inc.2025-03-04Adrian St. Clair Brownpending
TISSUE FACTOR ANTIBODY-DRUG CONJUGATES AND USES THEREOFA61K 47/6849, A61K 47/6889, A61K 47/68037, C07K 16/36Filed as EXELIXIS, INC.2025-02-25Robyn M. BARFIELDpending
METHODS FOR PROTEIN PURIFICATIONFiled as EXELIXIS, INC.2025-02-19LARRY JOE ANDERSONpending
C-MET MODULATOR PHARMACEUTICAL COMPOSITIONSA61K 31/47, A61K 9/00, A61K 9/2004, A61K 9/2009, A61K 9/2013, A61K 9/2018, A61K 9/2031, A61K 9/2054, A61K 9/2095, A61K 9/28, A61K 9/2833, A61K 9/2866, A61K 9/2893, A61K 31/00, A61K 31/33, A61K 31/395, A61K 31/435, A61K 45/06Filed as Exelixis, Inc.2025-01-02Jo Ann Wilsonpending
MALATE SALT OF N-(4-{[6,7-BIS(METHYLOXY) QUINOLIN-4-YL]OXY}PHENYL)-N'-(4-FLUOROPHENYL)CYCLOPROPANE-1,1-DICARBOXAMIDE, AND CRYSTALLINE FORMS THEREOF FOR THE TREATMENT OF CANCERA61K 31/47, C07D 215/22, C07D 215/233, A61P 43/00, A61P 25/00, A61P 5/14, A61P 35/00, C07B2200/13Filed as Exelixis, Inc.2024-11-25Adrian St. Clair Brown12275706
COMPOUNDS THAT INHIBIT POLO-LIKE KINASE 4Filed as EXELIXIS, INC.2024-11-19SANJAY BHATTARAIpending
5T4 ANTIBODY DRUG CONJUGATES AND METHODS OF THEIR USEFiled as EXELIXIS, INC.2024-11-14AMY PETERSONpending
COMPOUNDS THAT INHIBIT POLO-LIKE KINASE 4Filed as Exelixis, Inc.2024-11-08Brian Shererpending
METHODS FOR TREATING CANCER USING COMPOUNDS THAT INHIBIT PKMYT1Filed as EXELIXIS, INC.2024-11-07DANA GWINNpending
5T4 BINDING AGENTS AND USES THEREOFC07K 16/30, A61P 35/00, A61K2039/505, C07K2317/21, C07K2317/30, C07K2317/33, C07K2317/52, C07K2317/55, C07K2317/56, C07K2317/565, C07K2317/567, C07K2317/77, C07K2317/92, C07K2317/94, C07K2319/00Filed as EXELIXIS, INC.2024-11-06Bonnie HAMMERpending
5T4 ANTIBODY-DRUG CONJUGATES AND USES THEREOFA61K 47/6851, A61K 47/68031, C07K 16/30, A61K 47/6889, A61P 35/00, A61K 47/68033, A61K2039/505, C07K2317/21, C07K2317/33, C07K2317/34, C07K2317/55, C07K2317/92, C07K2317/94Filed as EXELIXIS, INC.2024-11-06Seema KANTAKpending
METHODS FOR TREATING CANCER USING COMPOUNDS THAT INHIBIT PKMYT1Filed as Exelixis, Inc.2024-10-04Dana GWINNpending
Processes for Preparing Quinoline Compounds and Pharmaceutical Compositions Containing Such CompoundsA61P 35/00, A61K 31/47, C07D 215/22, C07D 215/233Filed as Exelixis, Inc.2024-09-27Jo Ann Wilsonpending
ILT2 BINDING AGENTS AND USES THEREOFFiled as EXELIXIS, INC.2024-08-30RAMESH BALIGApending
ANTI-ROR ANTIBODY CONSTRUCTSA61P 35/00, C07K 16/2803, A61K 45/06, A61K2039/505, C07K 16/2809, C07K 16/2818, C07K 16/2878, C07K 16/468, C07K2317/24, C07K2317/31, C07K2317/35, C07K2317/522, C07K2317/524, C07K2317/526, C07K2317/55, C07K2317/77, C07K2317/92, C07K2317/94Filed as EXELIXIS, INC.2024-08-12Lucas BAILEYpending
MULTISPECIFIC BINDING AGENTS AND USES THEREOFC07K 16/2803, C07K 16/2827, A61K 47/6849, A61K 47/6879, A61P 35/00, A61K2039/505, A61K2039/545, C07K2317/31, C07K2317/73, C07K2317/732, C07K2317/76, C07K2317/92Filed as EXELIXIS, INC.2024-08-07Bryan GLASERpending
FUSED BICYCLIC HETEROCYCLYL COMPOUNDS AS USP1 INHIBITORSC07D 471/04, A61P 35/02, A61P 35/00, C07D 475/00, C07D 487/04, C07D 498/04, C07D 519/00Filed as Exelixis, Inc.2024-07-31Chandrasekhar ABBINENIpending
METHODS OF USE OF AGENTS THAT BIND TO NKG2A AND PD-L1Filed as EXELIXIS, INC.2024-07-31Seema KANTAKpending
TYROSINE-PROTEIN KINASE MEMBRANE RECEPTOR 1 (ROR1) ANTIBODY-DRUG CONJUGATES AND USES THEREOFFiled as EXELIXIS, INC.2024-07-19KATHLEEN GOGASpending
INTERLEUKIN-13 RECEPTOR SUBUNIT ALPHA-2 BINDING AGENTS AND USES THEREOFFiled as EXELIXIS, INC.2024-07-19RAMESH BALIGApending
PHARMACEUTICAL COMPOSITIONS COMPRISING ANTI-TISSUE FACTOR ANTIBODY-DRUG CONJUGATESA61K 47/6849, A61K 47/68031, A61K 47/6889, A61K 47/6851, A61P 35/00, A61K 9/0019, A61K 9/19, A61K 47/183, A61K 47/22, A61K 47/26Filed as EXELIXIS, INC.2024-07-19Mark REYNOLDSpending
ACTIVATABLE TYROSINE-PROTEIN KINASE MEMBRANE RECEPTOR (ROR) ANTIBODY-DRUG CONJUGATES AND USES THEREOFFiled as EXELIXIS, INC.2024-07-19MAXINE BAUZONpending
ACTIVATABLE ROR BINDING AGENTS AND USES THEREOFFiled as EXELIXIS, INC.2024-07-19FANGYONG DUpending
INTERLEUKIN-13 RECEPTOR SUBUNIT ALPHA-2 ANTIBODY-DRUG CONJUGATES AND USES THEREOFFiled as EXELIXIS, INC.2024-07-19PENELOPE M. DRAKEpending
FUSED PYRAZOLE DERIVATIVES AS USP1 INHIBITORSFiled as EXELIXIS, INC.2024-07-02CHANDRASEKHAR ABBINENIpending
CRYSTALLINE FORMS AND SALT FORMS OF A KINASE INHIBITORC07D 215/48, A61P 35/00Filed as Exelixis, Inc.2024-06-21Kirsten PHIZACKERLEYpending
METHOD OF TREATING CANCER AND BONE CANCER PAINA61K 31/47, A61K 31/517, C07D 215/233, A61P 19/00, A61P 25/04, A61P 35/04, A61P 35/00, A61K 31/536Filed as Exelixis, Inc.2024-06-04Gisela Schwabpending
MEK INHIBITORS AND METHODS OF THEIR USEA61K 31/397, C07D 205/04, C07D 205/06, C07D 403/06, A61P 17/06, A61P 43/00, A61P 35/02, A61P 17/02, A61P 35/00, C07D 401/04, C07D 401/06, C07D 401/12, C07D 401/14, C07D 403/04, C07D 403/12, C07D 405/12, C07D 409/06, C07D 409/12, C07D 413/12, C07D 413/14, C07D 417/12, C07D 471/04Filed as Exelixis, Inc.2024-05-23Naing Aaypending
Liquid Dosage Forms to Treat CancerA61K 31/47, A61P 35/00, A61K 9/0053Filed as Exelixis, Inc.2024-05-10Khalid Shahpending
CRYSTALLINE FORMS AND SALT FORMS OF A KINASE INHIBITORC07D 215/48, A61P 35/00, A61K 31/47, C07B2200/13Filed as Exelixis, Inc.2024-05-07Frenel DeMorin12679809
COMPOUNDS FOR THE TREATMENT OF KINASE-DEPENDENT DISORDERSC07D 215/48, A61K 31/47Filed as Exelixis, Inc.2024-05-02Khalid SHAHpending
METABOLITES OF N-(4-{[6,7-BIS(METHYLOXY)QUINOLIN-4-YL]OXY}PHENYL)-N'-(4-FLUOROPHENYL)CYCLOPROPANE-1,1-DICARBOXAMIDEC07C 233/60, C07D 215/22, C07C2601/02, A61P 35/00, C07C 305/24, C07D 215/60, G01N 33/487, G01N2570/00Filed as Exelixis, Inc.2024-04-22Dana T. Aftabpending
METHODS FOR TREATING CANCER USING COMPOUNDS THAT INHIBIT PKMYT1Filed as Exelixis, Inc.2024-04-05Dana Gwinnpending
AMHRII ANTIBODY-DRUG CONJUGATES AND USES THEREOFFiled as EXELIXIS, INC.2024-03-28YUTAKA MATSUDApending
Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms thereof for the treatment of cancerA61K 31/47, C07D 215/22, C07D 215/233, A61P 43/00, A61P 25/00, A61P 5/14, A61P 35/00, C07B2200/13Filed as Exelixis, Inc.2024-03-21Adrian St. Clair Brownpending
DLL3 ANTIBODY-DRUG CONJUGATES AND USES THEREOFFiled as EXELIXIS, INC.2024-03-21KATHLEEN GOGASpending
PROCESSES FOR PREPARING QUINOLINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH COMPOUNDSA61P 35/00, A61K 31/47, C07D 215/22, C07D 215/233Filed as Exelixis, Inc.2024-02-08Jo Ann Wilson12128039

Filings are matched to the company by applicant name, so a subsidiary filing under its own name is only here if that name resolves to this company. The applicant is printed as filed, which makes a wrong match visible. A patent is not a product: most applications are never granted, and most grants are never built.

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